SCHEMBL4540841

SCHEMBL4540841

O=c1[nH]n(Cc2ccc(F)cc2Cl)c2ccc(NS(=O)(=O)c3cccc4ccccc34)cc12

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.47
HTR6 P50406 10/20 0.42
P2RX7 Q99572 1/20 0.42
BRD4 O60885 3/20 0.41
FABP4 P15090 1/20 0.41
FABP5 Q01469 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
PFKFB3 Q16875 1/20 0.40
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN5 P54829 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1818816 0.89 PTGES2 (0.42) HTR6P2RX7BRD4ALDH1A1
SCHEMBL4536214 0.89 NR1I2 (0.52) NR1I2HTR6BRD4ALDH1A1HTT
SCHEMBL3903978 0.88 GSPT1 (0.41) NR1I2HTR6P2RX7BRD4PFKFB3
SCHEMBL4540174 0.84 NR1I2 (0.52) NR1I2HTR6BRD4ALDH1A1HTT
SCHEMBL1831975 0.82 GSPT1 (0.40) NR1I2HTR6P2RX7BRD4ALDH1A1
SCHEMBL3906145 0.79 MAP2K4 (0.39) BRD4ALDH1A1HTTHDAC1
SCHEMBL3907047 0.79 BRAF (0.44) HDAC1
SCHEMBL3918595 0.78 GSPT1 (0.42) NR1I2BRD4ALDH1A1
SCHEMBL1810508 0.78 NR1I2 (0.48) NR1I2HTR6BRD4FABP4FABP5
SCHEMBL3907924 0.77 TP53 (0.44) PTPN2PTPN1PTPN5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797042-B1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-01-07 EP claimed