SCHEMBL454160

SCHEMBL454160

O=C(O)c1ccc2c(c1)CC(Nc1ccc([N+](=O)[O-])cn1)CC2

nearest known ligand 0.81

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 9/20 0.81
HDAC6 Q9UBN7 4/20 0.50
HCAR3 P49019 5/20 0.47
SMN1; SMN2 Q16637 3/20 0.43
GAA P10253 2/20 0.43
NPC1 O15118 2/20 0.43
MAPT P10636 2/20 0.43
RAB9A P51151 2/20 0.43
CYP1A2 P05177 1/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL443904 0.90 HDAC8 (1.00) HDAC8HDAC6
SCHEMBL443905 0.78 HDAC8 (0.56) HDAC8HCAR3SMN1; SMN2GAANPC1
SCHEMBL456939 0.78 HDAC8 (0.79) HDAC8HDAC6
SCHEMBL2793284 0.75 GAA (0.58) HDAC8HCAR3SMN1; SMN2GAANPC1
SCHEMBL3318993 0.74 HDAC8 (0.56) HDAC8SMN1; SMN2GAANPC1MAPT
SCHEMBL444505 0.74 HDAC8 (1.00) HDAC8HDAC6
SCHEMBL2789965 0.72 MAPT (0.55) HDAC8HCAR3SMN1; SMN2GAAMAPT
SCHEMBL2789608 0.72 LMNA (0.59) HDAC8HCAR3SMN1; SMN2GAAMAPT
SCHEMBL8177053 0.72 GRIN2B (0.57) HDAC8GAANPC1MAPTRAB9A
SCHEMBL15680661 0.72 HDAC8 (0.71) HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2613775-A1 NOVEL N-HYDROXY-BENZAMIDES FOR THE TREATMENT OF CANCER F.HOFFMANN-LA ROCHE AG (CH) 2013-07-17 EP claimed
WO-2012031993-A1 NOVEL N-HYDROXY-BENZAMIDES FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2012-03-15 WO claimed