SCHEMBL4542407

SCHEMBL4542407

COC(=O)C1(CI)CCN(C(=O)OC(C)(C)C)CC1.[Li]CCCC

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
USP2 O75604 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TLR8 Q9NR97 1/20 0.36
EPHX2 P34913 1/20 0.34
GPR119 Q8TDV5 2/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
MMP13 P45452 3/20 0.34
ADAM17 P78536 3/20 0.34
MMP2 P08253 2/20 0.34
MMP14 P50281 1/20 0.34
EPHX1 P07099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4129353 0.89 PKM (0.48) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL27236283 0.81 PKM (0.44) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL6188518 0.81 USP2 (0.42) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL21963889 0.80 PKM (0.47) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL3970403 0.80 PKM (0.49) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL17020479 0.80 PKM (0.44) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL16986998 0.77 PKM (0.49) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL4295685 0.77 PKM (0.49) PKMCYP4F2CYP4A11USP2SMN1; SMN2
SCHEMBL3960309 0.77 CYP2D6 (0.46) USP2
SCHEMBL8263471 0.76 PKM (0.41) PKMCYP4F2CYP4A11USP2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013197-A1 PHENETHANOLAMINE DERIVATIVES AS BETA2 ADRENORECEPTOR AGONISTS AstraZeneca AB (SE) 2009-01-14 EP disclosed
WO-2007102771-A1 PHENETHANOLAMINE DERIVATIVES AS BETA2 ADRENORECEPTOR AGONISTS ASTRAZENECA AB (SE) 2007-09-13 WO disclosed