SCHEMBL4549142

SCHEMBL4549142

CC#Cc1cncc(-c2csc([C@]3(C)CC(=O)N(C)C(=NC(=O)OC(C)(C)C)N3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.54
CTSD P07339 9/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8258245 1.00 BACE1 (0.54) BACE1CTSD
SCHEMBL16480325 1.00 BACE1 (0.54) BACE1CTSD
SCHEMBL8436759 0.89 BACE1 (0.40) BACE1
SCHEMBL12916850 0.81 BACE1 (0.44) BACE1CTSD
SCHEMBL8247675 0.81 BACE1 (0.44) BACE1CTSD
SCHEMBL12172351 0.80 BACE1 (0.64) BACE1CTSD
SCHEMBL4549145 0.80 BACE1 (0.64) BACE1CTSD
SCHEMBL2948975 0.78 HCAR3 (0.32)
SCHEMBL2948973 0.78 HCAR3 (0.32)
SCHEMBL2948978 0.78 HCAR3 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168641-B2 Aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-01 US disclosed