SCHEMBL4549264

SCHEMBL4549264

CC#Cc1cncc(-c2sc([C@]3(C)CC(=O)N(C)C(=N)N3)cc2-c2cccnc2)c1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.45
CTSD P07339 3/20 0.33
CYP19A1 P11511 2/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
CYP17A1 P05093 1/20 0.32
CYP1A2 P05177 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
CYP3A4 P08684 1/20 0.32
GRM5 P41594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4549218 0.92 BACE1 (0.47) BACE1CTSDBACE2
SCHEMBL10186918 0.89 BACE1 (0.37) BACE1CTSDCYP19A1CYP11B1CYP11B2
SCHEMBL4549171 0.85 BACE1 (0.51) BACE1CTSDBACE2
SCHEMBL7560586 0.84 BACE1 (0.46) BACE1CTSDBACE2
SCHEMBL4549211 0.83 BACE1 (0.49) BACE1CTSDBACE2
SCHEMBL4549158 0.82 BACE1 (0.45) BACE1CTSDBACE2
SCHEMBL7553294 0.81 BACE1 (0.64) BACE1CTSDBACE2
SCHEMBL8436781 0.81 CYP11B2 (0.33) BACE1CYP11B1CYP11B2
SCHEMBL7570060 0.80 BACE1 (0.40) BACE1CTSDCYP19A1CYP11B1CYP11B2
SCHEMBL4549143 0.79 BACE1 (0.48) BACE1CTSDBACE2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168641-B2 Aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-01 US disclosed