SCHEMBL4549702

SCHEMBL4549702

COc1cc(CC(=O)O)c(Cl)cc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.53
HSD17B10 Q99714 1/20 0.47
NPSR1 Q6W5P4 1/20 0.43
CYP3A4 P08684 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CXCL8 P10145 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
SELP P16109 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3323483 0.86 HSD17B10 (0.53) GAAHSD17B10NPSR1CYP3A4ALDH1A1
SCHEMBL16068896 0.85 HSD17B10 (0.51) GAAHSD17B10NPSR1CYP3A4ALDH1A1
SCHEMBL19180928 0.83 GAA (0.49) GAACYP3A4ALDH1A1NPC1TSHR
SCHEMBL2729269 0.82 GAA (0.53) GAAHSD17B10NPSR1CYP3A4ALDH1A1
SCHEMBL2124489 0.81 HSD17B10 (0.51) GAAHSD17B10NPSR1CYP3A4ALDH1A1
SCHEMBL7714917 0.81 GAA (0.54) GAAHSD17B10CYP3A4ALDH1A1NPC1
SCHEMBL5373257 0.81 HSD17B10 (0.47) GAAHSD17B10NPSR1CYP3A4ALDH1A1
SCHEMBL3918194 0.81 HSD17B10 (0.47) GAAHSD17B10NPSR1CYP3A4ALDH1A1
SCHEMBL19175614 0.80 GAA (0.60) GAAHSD17B10CYP3A4ALDH1A1NPC1
SCHEMBL3580327 0.79 GAA (0.48) GAACXCL8CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058134-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed