SCHEMBL4549816

SCHEMBL4549816

C[C@@H]1CN(c2ccc(N)nc2)CCO1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.43
CCND1 P24385 1/20 0.43
CDK6 Q00534 1/20 0.43
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
PIK3CA P42336 3/20 0.41
MTOR P42345 3/20 0.41
PIK3R1 P27986 2/20 0.41
LRRK2 Q5S007 5/20 0.40
FFAR2 O15552 4/20 0.40
GAK O14976 3/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21698724 1.00 CDK4 (0.43) CDK4CCND1CDK6MAPTRAB9A
SCHEMBL17340556 1.00 CDK4 (0.43) CDK4CCND1CDK6MAPTRAB9A
SCHEMBL2722889 0.83 MAPT (0.58) CDK4CCND1CDK6MAPTRAB9A
SCHEMBL4825445 0.83 MAPT (0.58) CDK4CCND1CDK6MAPTRAB9A
SCHEMBL28876591 0.82 PIK3CA (0.40) CDK4CCND1CDK6MAPTPIK3CA
SCHEMBL28076420 0.82 PIK3CA (0.40) PIK3CAMTORPIK3R1CHRNB2CHRNA4
SCHEMBL28876546 0.81 PIK3CA (0.37) MAPTPIK3CAMTORPIK3R1CHRNB2
SCHEMBL14167561 0.81 MAPT (0.46) CDK4CCND1CDK6MAPTRAB9A
SCHEMBL12236694 0.81 MAPT (0.46) CDK4CCND1CDK6MAPTRAB9A
SCHEMBL23104529 0.79 ADORA2A (0.49) PIK3CAMTORPIK3R1LRRK2CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061156-A1 CDK INHIBITORS TAVARES FRANCIS X (US) 2012-05-10 WO disclosed