SCHEMBL4550316

SCHEMBL4550316

CC(=O)Nc1cc(C(=O)NC(C)c2cnc(OCC(F)(F)F)c(CI)c2)ccn1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.50
MAPT P10636 5/20 0.50
ACACB O00763 4/20 0.45
SCN9A Q15858 1/20 0.43
GSK3A P49840 3/20 0.42
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 3/20 0.38
AAK1 Q2M2I8 3/20 0.38
ROCK2 O75116 3/20 0.37
FDPS P14324 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4550821 0.93 GSK3B (0.59) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL4550508 0.91 GSK3B (0.49) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2713653 0.88 GSK3B (0.50) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2716385 0.88 GSK3B (0.50) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2716135 0.88 SCN9A (0.52) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2715577 0.87 GSK3B (0.51) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2718053 0.85 GSK3B (0.60) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2713575 0.83 ACACB (0.50) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL18266121 0.82 GSK3B (0.45) GSK3BMAPTACACBSCN9AGSK3A
SCHEMBL2713908 0.82 GSK3B (0.61) GSK3BMAPTACACBSCN9AGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed