SCHEMBL4550351

SCHEMBL4550351

Bc1cc(CNC(=O)c2ccnc(NC(=O)C3CC3)n2)cnc1OCC(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 10/20 0.45
GSK3A P49840 8/20 0.45
JAK1 P23458 2/20 0.38
AURKA O14965 2/20 0.37
SYK P43405 2/20 0.37
LCK P06239 1/20 0.37
IGF1R P08069 1/20 0.37
EIF2AK2 P19525 1/20 0.37
BMX P51813 1/20 0.37
MAPT P10636 2/20 0.37
KLKB1 P03952 1/20 0.37
JAK2 O60674 2/20 0.36
CNR2 P34972 1/20 0.34
ABL1 P00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2716932 0.90 GSK3B (0.45) GSK3BGSK3AJAK1AURKASYK
SCHEMBL2716154 0.90 GSK3B (0.47) GSK3BGSK3AAURKASYKLCK
SCHEMBL2716231 0.90 GSK3B (0.45) GSK3BGSK3AAURKASYKLCK
SCHEMBL2716708 0.90 GSK3B (0.45) GSK3BGSK3AJAK1AURKASYK
SCHEMBL2718565 0.89 GSK3B (0.44) GSK3BGSK3AJAK1AURKASYK
SCHEMBL2715923 0.88 GSK3B (0.44) GSK3BGSK3ASYKIGF1RCNR2
SCHEMBL4550343 0.84 GSK3B (0.60) GSK3BGSK3AMAPT
SCHEMBL2713486 0.84 KLKB1 (0.46) GSK3BGSK3ASYKKLKB1
SCHEMBL2713402 0.82 GSK3B (0.37) GSK3BGSK3AJAK1SYKMAPT
SCHEMBL2716643 0.80 ALDH1A1 (0.43) GSK3BGSK3AJAK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed