SCHEMBL4550698

SCHEMBL4550698

NC(CC(=O)N1CCc2cnc(C(F)(F)F)nc2C1)Cc1cc(F)c(F)cc1F

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.61
DPP8 Q6V1X1 11/20 0.61
DPP7 Q9UHL4 7/20 0.61
DPP9 Q86TI2 6/20 0.55
ACE P12821 1/20 0.55
HTR2A P28223 1/20 0.55
FAP Q12884 1/20 0.55
CYP3A4 P08684 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4550697 1.00 DPP4 (0.61) DPP4DPP8DPP7DPP9ACE
Hydrochloric Acid SCHEMBL4399414 0.99 DPP4 (0.61) DPP4DPP8DPP7DPP9ACE
SCHEMBL8345171 0.90 DPP4 (0.66) DPP4DPP8DPP7DPP9
SCHEMBL4387254 0.86 DPP4 (0.56) DPP4DPP8DPP7DPP9
SCHEMBL4392074 0.82 DPP4 (0.44) DPP4DPP8DPP7DPP9ACE
SCHEMBL4400632 0.77 DPP4 (0.60) DPP4DPP8DPP7DPP9
SCHEMBL5228197 0.76 DPP4 (1.00) DPP4DPP8DPP7DPP9ACE
Hydrochloric Acid SCHEMBL4399397 0.76 DPP4 (0.59) DPP4DPP8DPP7DPP9
Hydrochloric Acid SCHEMBL1842316 0.76 DPP4 (0.98) DPP4DPP8DPP7DPP9ACE
SCHEMBL16161427 0.75 DPP4 (0.72) DPP4DPP8DPP7DPP9ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554256-B1 PIPERIDINO PYRIMIDINE DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OF DIABETES MERCK & CO INC (US) 2009-12-09 EP disclosed