SCHEMBL4550806

SCHEMBL4550806

CC(=O)Nc1cc(C(=O)NCc2cnc(OCC(F)(F)F)c(CI)c2)ccn1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 6/20 0.47
MAPT P10636 4/20 0.47
SCN9A Q15858 1/20 0.44
GSK3A P49840 3/20 0.43
KCNH2 Q12809 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
GRK2 P25098 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
RIPK1 Q13546 3/20 0.38
HTT P42858 2/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM1A O60341 1/20 0.37
HDAC1 Q13547 1/20 0.37
EPHX2 P34913 3/20 0.37
ALDH1A1 P00352 1/20 0.37
ROS1 P08922 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2718782 0.93 GSK3B (0.51) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL4550807 0.91 GSK3B (0.46) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL2715052 0.88 GSK3B (0.47) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL2715625 0.88 GSK3B (0.47) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL2716945 0.87 SCN9A (0.54) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL2715374 0.87 GSK3B (0.47) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL2719835 0.86 GSK3B (0.48) GSK3BMAPTSCN9AGSK3AL3MBTL1
SCHEMBL2716722 0.85 GSK3B (0.47) GSK3BMAPTSCN9AGSK3AGRK2
SCHEMBL2716288 0.84 GSK3B (0.61) GSK3BMAPTSCN9AGSK3AKCNH2
SCHEMBL2714719 0.84 GSK3B (0.50) GSK3BMAPTSCN9AGSK3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed