SCHEMBL4550972

SCHEMBL4550972

CC(=O)c1sccc1NS(=O)(=O)c1ccc(C2CCCC2)cc1F

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.54
PIK3C3 Q8NEB9 2/20 0.40
NRP1 O14786 1/20 0.40
SCN9A Q15858 5/20 0.39
PARP14 Q460N5 1/20 0.39
SLC10A6 Q3KNW5 1/20 0.39
WDR5 P61964 1/20 0.37
LMNA P02545 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KDM1A O60341 1/20 0.37
ACLY P53396 1/20 0.37
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
CCR2 P41597 2/20 0.36
SCN1A P35498 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN8A Q9UQD0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2748477 0.90 KCNH2 (0.53) KCNH2PIK3C3NRP1SCN9APARP14
SCHEMBL2748212 0.90 KCNH2 (0.70) KCNH2PARP14SLC10A6LMNAALDH1A1
SCHEMBL4547553 0.82 KCNH2 (0.43) KCNH2PIK3C3NRP1SCN9AWDR5
SCHEMBL2747486 0.73 KCNH2 (0.53) KCNH2NRP1PARP14WDR5KDM4E
SCHEMBL2747534 0.73 KCNH2 (0.70) KCNH2PARP14SLC10A6LMNAKDM4E
SCHEMBL1199270 0.71 KCNH2 (1.00) KCNH2NRP1PARP14SLC10A6LMNA
SCHEMBL2747281 0.71 KDM1A (0.55) LMNAKDM4EALDH1A1KDM1AACLY
SCHEMBL2748805 0.70 LMNA (0.67) KCNH2SLC10A6LMNAKDM4EALDH1A1
SCHEMBL1199591 0.70 KCNH2 (0.80) KCNH2PARP14SLC10A6LMNAALDH1A1
SCHEMBL2748631 0.70 KCNH2 (0.60) KCNH2NRP1PARP14SLC10A6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178699-B2 Modulators of CCR9 receptor and methods of use thereof PFIZER INC. (US) 2012-05-15 US disclosed
US-20100029753-A1 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. 2010-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029753-A1 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF CCR9, CCR1, CCR4 KCNH2 4765/4885PIK3C3 3160/4885NRP1 543/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.