SCHEMBL4551133

SCHEMBL4551133

O=C(F)c1cc2ccccc2n1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.51
MCL1 Q07820 1/20 0.50
ALDH1A1 P00352 2/20 0.49
TSHR P16473 1/20 0.49
CCR2 P41597 4/20 0.45
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
PLA2G10 O15496 1/20 0.40
NOD2 Q9HC29 1/20 0.40
NOD1 Q9Y239 1/20 0.40
SLC9A1 P19634 1/20 0.40
MAPT P10636 1/20 0.39
LDHA P00338 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PDGFRB P09619 1/20 0.38
KDR P35968 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3638561 0.85 DAO (0.65) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL29780995 0.85 DAO (0.65) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL28160836 0.82 PLA2G10 (0.54) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL3843739 0.78 DAO (0.46) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL4467286 0.76 DAO (0.47) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL5967722 0.74 MCL1 (0.49) DAOMCL1ALDH1A1TSHRCYP1A2
SCHEMBL30343692 0.74 MCL1 (0.49) DAOMCL1ALDH1A1TSHRCYP1A2
SCHEMBL3842692 0.74 DAO (0.46) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL17422801 0.74 DAO (0.46) DAOMCL1ALDH1A1TSHRCCR2
SCHEMBL3672379 0.74 DAO (0.42) DAOMCL1ALDH1A1TSHRCCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010535-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120098-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed