SCHEMBL4551203

SCHEMBL4551203

Cc1ccc(NC(=O)c2cccc(F)c2)cc1-c1cc(C(=O)NCC(C)(C)C)on1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
BRAF P15056 9/20 0.45
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
CTDSP1 Q9GZU7 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 3/20 0.44
KDM4E B2RXH2 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RAF1 P04049 8/20 0.43
TP53 P04637 1/20 0.43
CASP3 P42574 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
DYRK3 O43781 1/20 0.42
ROCK2 O75116 1/20 0.42
MAP4K4 O95819 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417419 0.91 GLA (0.48) BRAFRAF1
SCHEMBL4407858 0.89 RAF1 (0.55) BRAFRAF1
SCHEMBL4565727 0.89 NR1H4 (0.48) BRAFRAF1
SCHEMBL4408307 0.89 RAF1 (0.42) BRAFRAF1
SCHEMBL4565699 0.89 BRAF (0.45) CYP1A2CYP2C19BRAFKCNK3KCNK9
SCHEMBL4565940 0.88 FFAR1 (0.46) CYP1A2CYP2C19BRAFNPC1RAF1
SCHEMBL4565578 0.88 RAF1 (0.46) BRAFRAF1
SCHEMBL4551200 0.88 CSGALNACT1 (0.44) CYP1A2CYP2C19BRAFNPC1RAB9A
SCHEMBL4413519 0.88 HSP90AA1 (0.49) CYP1A2CYP2C19BRAFKCNK3KCNK9
SCHEMBL4565554 0.88 BRAF (0.47) BRAFRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035005-A2 THERAPY USING CYTOKINE INHIBITORS Kemia, INC. (US) 2009-03-18 EP disclosed
WO-2007146712-A2 THERAPY USING CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-12-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed