SCHEMBL4552114

SCHEMBL4552114

C#Cc1cccc2c1OCCO2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.44
ICAM1 P05362 1/20 0.44
ITGAL P20701 1/20 0.44
ADRB1 P08588 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 3/20 0.40
CRHBP P24387 2/20 0.40
CRHR2 Q13324 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 1/20 0.40
MTNR1A P48039 4/20 0.38
EGFR P00533 1/20 0.37
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTR1A P08908 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
PMP22 Q01453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5612838 0.84 ABCG2 (0.44) KDM4ELMNABRD4CREBBPALDH1A1
SCHEMBL97610 0.80 KDM4E (0.45) ITGB2ICAM1ITGALADRB1KDM4E
SCHEMBL7128137 0.80 ITGB2 (0.44) ITGB2ICAM1ITGALADRB1KDM4E
SCHEMBL18936123 0.76 BRD4 (0.33) BRD4CREBBP
SCHEMBL21160350 0.74 PARP1 (0.47) BRD4CREBBP
SCHEMBL3787577 0.72 ITGB2 (0.50) ITGB2ICAM1ITGALADRB1KDM4E
SCHEMBL1663066 0.72 ITGB2 (0.50) ITGB2ICAM1ITGALADRB1KDM4E
SCHEMBL3072409 0.72 ITGB2 (0.55) ITGB2ICAM1ITGALADRB1KDM4E
SCHEMBL18936074 0.69 BRD4 (0.33) BRD4CREBBP
SCHEMBL24312061 0.68 ITGB2 (0.50) ITGB2ICAM1ITGALADRB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299354-B1 FACTOR VIIA INHIBITORY (THIO)UREA DERIVATIVES, THEIR PREPARATION AND THEIR USE SANOFI AVENTIS DEUTSCHLAND (DE) 2009-07-22 EP claimed