SCHEMBL4552394

SCHEMBL4552394

COC1C=c2[nH]c(CNC(O)(CC(C)CF)C(F)F)cc2=CN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3699945 0.83
SCHEMBL4552393 0.79
SCHEMBL6381722 0.71
SCHEMBL4431839 0.68 CASR (0.43)
SCHEMBL3817481 0.65 NR3C1 (0.39)
SCHEMBL3825741 0.65
SCHEMBL3826673 0.65 NR3C1 (0.39)
SCHEMBL21728189 0.46
SCHEMBL21728185 0.43
SCHEMBL21211591 0.42

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121670-A2 SYNTHESIS OF SELECTED STEREOISOMERS OF CERTAIN SUBSTITUTED ALCOHOLS Bausch & Lomb Incorporated (US) 2009-11-25 EP disclosed
WO-2008088969-A2 SYNTHESIS OF SELECTED STEREOISOMERS OF CERTAIN SUBSTITUTED ALCOHOLS BAUSCH & LOMB INCORPORATED (US) 2008-07-24 WO disclosed