SCHEMBL4553386

SCHEMBL4553386

Nc1nccc(-c2c[nH]cc2C#Cc2ccccc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.52
CDK5 Q00535 8/20 0.47
CDK5R1 Q15078 8/20 0.47
GSK3B P49841 7/20 0.47
DYRK1A Q13627 6/20 0.47
CLK1 P49759 3/20 0.47
MAP3K14 Q99558 2/20 0.47
PRKACA P17612 3/20 0.46
AURKA O14965 1/20 0.46
HSP90AA1 P07900 1/20 0.46
ADORA2A P29274 1/20 0.46
NFATC1 O95644 2/20 0.43
CCNT1 O60563 4/20 0.43
CCNA2 P20248 4/20 0.43
CDK2 P24941 4/20 0.43
CDK9 P50750 4/20 0.43
CCNA1 P78396 4/20 0.43
PDPK1 O15530 2/20 0.43
CCNB2 O95067 2/20 0.40
CDK1 P06493 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2993571 0.79 CDK5 (0.58) GRM4CDK5CDK5R1GSK3BDYRK1A
SCHEMBL10338425 0.70 GRM4 (1.00) GRM4PRKACAAURKAHSP90AA1ADORA2A
SCHEMBL18130895 0.66 HSP90AA1 (0.60) GRM4CDK5CDK5R1GSK3BDYRK1A
SCHEMBL30046927 0.66 HSP90AA1 (0.60) GRM4CDK5CDK5R1GSK3BDYRK1A
SCHEMBL1388378 0.65 DHFR (0.54) GRM4ADORA2A
SCHEMBL316210 0.65 HSP90AA1 (1.00) GRM4GSK3BPRKACAAURKAHSP90AA1
SCHEMBL573402 0.64 GSK3B (1.00) CDK5CDK5R1GSK3BDYRK1ACLK1
SCHEMBL29488162 0.64 GSK3B (1.00) CDK5CDK5R1GSK3BDYRK1ACLK1
Hydrochloric Acid SCHEMBL17186384 0.64 HSP90AA1 (0.96) GRM4GSK3BPRKACAAURKAHSP90AA1
SCHEMBL5140478 0.63 FEN1 (0.57) GRM4CDK5CDK5R1GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125803-A1 PYRROLO[2,3-B]PYRIDINE COMPOUNDS, AZAINDOLE COMPOUNDS USED FOR SYNTHESIZING SAID PYRROLO[2,3-B]PYRIDINE COMPOUNDS, METHODS FOR THE PRODUCTION THEREOF, AND USES THEREOF Centre National de la Recherche Scientifique (FR) 2009-12-02 EP disclosed
WO-2008129152-A1 PYRROLO[2,3-B]PYRIDINE COMPOUNDS, AZAINDOLE COMPOUNDS USED FOR SYNTHESIZING SAID PYRROLO[2,3-B]PYRIDINE COMPOUNDS, METHODS FOR THE PRODUCTION THEREOF, AND USES THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2008-10-30 WO disclosed