Vorozole

Vorozole

SCHEMBL4554

Cn1nnc2ccc([C@H](c3ccc(Cl)cc3)n3cncn3)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 20/20 1.00
CYP11B1 P15538 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rac-Vorozole SCHEMBL13223107 1.00 CYP19A1 (1.00) CYP19A1CYP11B1
Vorozole SCHEMBL29363602 1.00 CYP19A1 (1.00) CYP19A1CYP11B1
[N-Methyl-11C]Vorozole SCHEMBL12171619 1.00 CYP19A1 (1.00) CYP19A1CYP11B1
Rac-Vorozole SCHEMBL29606650 1.00 CYP19A1 (1.00) CYP19A1CYP11B1
Rac-Vorozole SCHEMBL1552681 1.00 CYP19A1 (1.00) CYP19A1CYP11B1
Vorozole SCHEMBL19127035 0.92 CYP19A1 (0.84) CYP19A1CYP11B1
SCHEMBL13223109 0.91 CYP19A1 (0.83) CYP19A1CYP11B1
SCHEMBL13223108 0.91 CYP19A1 (0.83) CYP19A1CYP11B1
SCHEMBL3871739 0.86 CYP19A1 (0.76) CYP19A1CYP11B1
Oxalic Acid SCHEMBL9524494 0.84 CYP19A1 (0.72) CYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 30870 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-3645742-B1 ANTI-ROR1 ANTIBODIES AND METHODS OF MAKING AND USING THEREOF SYSTIMMUNE INC (US) 2026-04-29 EP claimed
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2026-04-23 US claimed
US-20260103461-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF OLEMA PHARMACEUTICALS INC (US) 2026-04-16 US claimed
EP-4712980-A1 TREATMENT OF BREAST TISSUE Havah Therapeutics Pty Ltd (AU) 2026-03-25 EP claimed
US-12576077-B2 Composition for preventing, alleviating or treating cancer CKP THERAPEUTICS, INC. (US) 2026-03-17 US claimed
EP-4680226-A2 ACYLSULFONAMIDE KAT6A INHIBITORS Olema Pharmaceuticals, Inc. (US) 2026-01-21 EP claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4653019-A1 ANTI-HER2 ANTIBODY-DRUG CONJUGATE FOR TREATING BREAST CANCER Jiangsu Hengrui Pharmaceuticals Co., Ltd. (CN) 2025-11-26 EP claimed
CN-1261803-A Antioxidant enhancement of therapy for hyperproliferative conditions ATHEROGENICS INC (US) 2000-08-02 CN claimed
WO-2000043553-A1 IDENTIFYING, MONITORING, AND TREATING WOMEN FOR BREAST PRECANCER OR CANCER PRO-DUCT HEALTH, INC. (US) 2000-07-27 WO claimed
EP-1019034-A2 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS Atherogenics, Inc. (US) 2000-07-19 EP claimed
US-6020327-A Control of hair growth THE CENTRAL SHEFFIELD UNIVERSITY HOSPITALS NHS TRUST (GB) 2000-02-01 US claimed
US-5972921-A UROGENITAL DISORDERS IN MALES HORMOS MEDICAL OY LTD. (FI) 1999-10-26 US claimed
WO-1999030708-A2 USE OF AN AROMATASE INHIBITOR IN THE TREATMENT OF DECREASED ANDROGEN TO ESTROGEN RATIO AND DETRUSOR URETHRAL SPHINCTER DYSSYNERGIA IN MEN AND METHOD TO STUDY THE DYSSYNERGIA IN MALE RODENTS HORMOS MEDICAL OY LTD. (FI) 1999-06-24 WO claimed
WO-1999001118-A9 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS ATHEROGENICS INC (US) 1999-05-20 WO claimed
US-5861389-A TREATING MALE MENOPAUSE SCHERING AKTIENGESELLSCHAFT (DE) 1999-01-19 US claimed
WO-1999001118-A2 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS ATHEROGENICS, INC. (US) 1999-01-14 WO claimed
WO-1997006788-A1 TRANSDERMAL ADMINISTRATION OF VOROZOLE JANSSEN PHARMACEUTICA N.V. (BE) 1997-02-27 WO claimed