SCHEMBL4555115

SCHEMBL4555115

CCCSc1nc(C(F)(F)F)ccc1/C=C/C(=O)O.O=C(O)/C=C/c1ccc(C(F)(F)F)nc1Cl

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 3/20 0.34
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ESR1 P03372 1/20 0.33
PPARG P37231 3/20 0.33
PPARD Q03181 3/20 0.33
TRPV1 Q8NER1 4/20 0.32
PPARA Q07869 2/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
MIF P14174 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555116 1.00 ALDH1A1 (0.34) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL3776850 0.93 ALDH1A1 (0.38) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL3776848 0.93 ALDH1A1 (0.38) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL4555117 0.89 TRPV1 (0.32) TRPV1
SCHEMBL3778281 0.84 ALDH1A1 (0.38) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL3778284 0.84 ALDH1A1 (0.38) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL3778055 0.83 MIF (0.41) ALDH1A1KDM4EGAAPPARGPPARD
SCHEMBL3783377 0.83 MIF (0.41) ALDH1A1KDM4EGAAPPARGPPARD
SCHEMBL13017803 0.74 TRPV1 (0.40) KDM4EKMT2ATRPV1LMNAMAPT
SCHEMBL3776043 0.74 MEN1 (0.38) ALDH1A1KDM4EGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054411-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST; AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2009-05-06 EP disclosed
WO-2008013414-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST; AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2008-01-31 WO disclosed