SCHEMBL4555746

SCHEMBL4555746

Clc1nc(N2CCOCC2)c2sc(C[N+]3(C4CCNCC4)CCCCC3)cc2n1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.42
PIK3R1 P27986 7/20 0.42
MTOR P42345 3/20 0.41
PIK3CD O00329 10/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4553952 0.85 SMN1; SMN2 (0.38) PIK3CAMTORSMN1; SMN2PIK3CBPIK3CG
SCHEMBL5252377 0.82 PIK3CA (0.61) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL1089140 0.76 PIK3CA (0.42) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL189736 0.76 PIK3CA (0.53) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL1181831 0.75 PIK3CA (0.43) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL4555688 0.75 PIK3CA (0.41) PIK3CAPIK3R1MTORPIK3CDSMN1; SMN2
SCHEMBL5251923 0.75 PIK3CA (0.41) PIK3CAPIK3R1MTORPIK3CDSMN1; SMN2
Hydrochloric Acid SCHEMBL30151144 0.75 PIK3CA (0.53) PIK3CAPIK3R1MTORPIK3CDPIK3CB
Hydrochloric Acid SCHEMBL1182606 0.75 PIK3CA (0.53) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL190175 0.74 PIK3CA (0.39) PIK3CAPIK3R1MTORPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114949-A1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND METHODS OF USE F.HOFFMANN-LA ROCHE AG (CH) 2009-11-11 EP disclosed
WO-2008070740-A1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND METHODS OF USE F.HOFFMANN-LA ROCHE AG (CH) 2008-06-12 WO disclosed