SCHEMBL4556713

SCHEMBL4556713

Cc1cccc(C)c1NC(=O)c1ccc(Nc2nc(S(C)(=O)=O)c3ccccc3n2)cc1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.45
HDAC3 O15379 1/20 0.45
APP P05067 1/20 0.45
ACHE P22303 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
TNKS O95271 1/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4154962 0.86 MAPT (0.54) PTGER4HDAC3APPACHEHDAC4
SCHEMBL4142299 0.83 MAPT (0.55) PTGER4MAPT
SCHEMBL4135480 0.82 MAPT (0.47) PTGER4HDAC3APPACHEHDAC4
SCHEMBL4129833 0.80 MERTK (0.46) PTGER4HDAC3APPACHEHDAC4
SCHEMBL4139018 0.80 LMNA (0.48) MAPT
SCHEMBL4566757 0.80
SCHEMBL4145093 0.79 LMNA (0.47) MAPT
SCHEMBL4132697 0.78 MERTK (0.48) PTGER4
SCHEMBL4148217 0.77 TNKS (0.51) TNKSMAPT
SCHEMBL4130005 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134695-A1 INHIBITORS OF THE HEDGEHOG PATHWAY Exelixis, Inc. (US) 2009-12-23 EP claimed
WO-2008112913-A1 INHIBITORS OF THE HEDGEHOG PATHWAY EXELIXIS, INC. (US) 2008-09-18 WO claimed