SCHEMBL4556961

SCHEMBL4556961

CC(C)(C)N1C(=O)C(O)(C(F)(F)F)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CHRM1 P11229 3/20 0.44
PDK2 Q15119 10/20 0.42
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RAD52 P43351 1/20 0.36
CNR1 P21554 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14101179 0.80 RAD52 (0.51) TSHRSMN1; SMN2CHRM1PDK2ALDH1A1
SCHEMBL16997509 0.78 MEN1 (0.37) TSHRSMN1; SMN2ALDH1A1NPSR1RAD52
Bromide SCHEMBL6851490 0.75 PGR (0.42) PDK2NPSR1
SCHEMBL31389172 0.70 RAD52 (0.51) TSHRSMN1; SMN2ALDH1A1RAD52
SCHEMBL16940892 0.67 KMT2A (0.43) TSHRALDH1A1NPSR1
SCHEMBL20229558 0.66 KDM4E (0.31)
SCHEMBL15203037 0.65 PDK2 (0.76) PDK2
SCHEMBL12536165 0.64 TSHR (0.47) TSHRSMN1; SMN2CHRM1PDK2ALDH1A1
SCHEMBL19319616 0.63 CNR1 (0.40) SMN1; SMN2CHRM1ALDH1A1NPSR1CNR1
SCHEMBL19654624 0.63 MEN1 (0.37) SMN1; SMN2PDK2CNR1GPR55TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2009502856-A 2009-01-29 JP claimed
EP-1915357-A1 2-HYDROXY-PROPIONIC ACID DERIVATIVES AND 3-HYDROXY-BENZOFURAN-2-ONE DERIVATIVES WITH AFFINITY FOR THE GABA-B-RECEPTOR F. Hoffmann-Roche AG (CH) 2008-04-30 EP claimed
WO-2007014843-A1 2-HYDROXY-PROPIONIC ACID DERIVATIVES AND 3-HYDROXY-BENZOFURAN-2-ONE DERIVATIVES WITH AFFINITY FOR THE GABA-B-RECEPTOR F. HOFFMANN-LA ROCHE AG (CH) 2007-02-08 WO claimed