SCHEMBL455795

SCHEMBL455795

CC(C(N)=O)c1ccc(C#Cc2ccc(O)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.50
APP P05067 4/20 0.47
FFAR1 O14842 1/20 0.42
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ACACB O00763 7/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1064971 0.89 EPHX1 (0.60) EPHX1APPESR1ESR2PDCD1
SCHEMBL458652 0.87 EPHX1 (0.51) EPHX1APPFFAR1ACACB
Hydrochloric Acid SCHEMBL15663072 0.87 EPHX1 (0.58) EPHX1APPESR1ESR2PDCD1
SCHEMBL456155 0.81 ACACB (0.60) EPHX1APPMAPTACACB
SCHEMBL455771 0.78 EPHX1 (0.53) EPHX1APPFFAR1ESR1
SCHEMBL462901 0.77 GAA (0.47) APPFFAR1GAAMAPTCRHBP
SCHEMBL18130044 0.77 APP (0.58) APPFFAR1ESR1ESR2PDCD1
SCHEMBL964721 0.72 EPHX1 (0.60) EPHX1APPESR1GAA
SCHEMBL16750533 0.72 EPHX1 (0.60) EPHX1APPSMN1; SMN2
SCHEMBL13446952 0.72 EPHX1 (0.60) EPHX1APPESR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614054-A1 ETHYNE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF Boehringer Ingelheim International GmbH (DE) 2013-07-17 EP disclosed
WO-2012032014-A1 ETHYNE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-03-15 WO disclosed