SCHEMBL458652

SCHEMBL458652

CC(C)c1ccc(C#Cc2ccc(C(C)C(N)=O)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.51
ACACB O00763 10/20 0.49
FFAR1 O14842 1/20 0.44
KIF11 P52732 1/20 0.42
HTT P42858 1/20 0.41
APP P05067 1/20 0.41
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HIF1A Q16665 1/20 0.38
ADK P55263 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455795 0.87 EPHX1 (0.50) EPHX1ACACBFFAR1APP
SCHEMBL456155 0.83 ACACB (0.60) EPHX1ACACBAPP
SCHEMBL8141103 0.79 ACACB (0.50) ACACBFFAR1HTTAPPADK
SCHEMBL455771 0.79 EPHX1 (0.53) EPHX1FFAR1APPCYP2C9
SCHEMBL964721 0.78 EPHX1 (0.60) EPHX1KIF11HTTAPPCYP2C9
SCHEMBL13446952 0.78 EPHX1 (0.60) EPHX1KIF11HTTAPPCYP2C9
SCHEMBL3261236 0.78 EPHX1 (0.60) EPHX1KIF11HTTAPPCYP2C9
SCHEMBL7794207 0.76 EPHX1 (0.58) EPHX1APPCYP2D6CYP2C9
SCHEMBL607802 0.76 EPHX1 (0.58) EPHX1APPCYP2D6CYP2C9
SCHEMBL607803 0.76 EPHX1 (0.58) EPHX1APPCYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614054-A1 ETHYNE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF Boehringer Ingelheim International GmbH (DE) 2013-07-17 EP disclosed
WO-2012032014-A1 ETHYNE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-03-15 WO disclosed