SCHEMBL4558241

SCHEMBL4558241

NCc1cc(N)ccc1O.Nc1ccc(N)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
CYP3A4 P08684 7/20 0.53
TSHR P16473 4/20 0.53
ALDH1A1 P00352 3/20 0.53
HPGD P15428 3/20 0.53
ALOX15 P16050 3/20 0.53
HSD17B10 Q99714 2/20 0.53
THRB P10828 2/20 0.53
CASP1 P29466 2/20 0.53
RECQL P46063 1/20 0.53
PRKCI P41743 1/20 0.46
ACHE P22303 3/20 0.45
ESR2 Q92731 1/20 0.41
MAPK1 P28482 2/20 0.38
ALOX12 P18054 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PDE10A Q9Y233 1/20 0.37
CA12 O43570 1/20 0.37
CA4 P22748 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL34055 0.85 PRKCI (0.59) CA1CA2CYP3A4TSHRALDH1A1
Hydrochloric Acid SCHEMBL1986970 0.83 ACHE (0.60) CA1CA2CYP3A4TSHRALDH1A1
Hydrochloric Acid SCHEMBL2480499 0.83 ACHE (0.60) CA1CA2CYP3A4TSHRALDH1A1
SCHEMBL11682542 0.78 PRKCI (0.49) CA1CA2CYP3A4TSHRALDH1A1
SCHEMBL33731 0.77
SCHEMBL29437149 0.77
Hydrochloric Acid SCHEMBL10882631 0.74 CYP3A4 (0.71) CA1CA2CYP3A4TSHRALDH1A1
Hydrochloric Acid SCHEMBL28886798 0.74 CYP3A4 (0.71) CA1CA2CYP3A4TSHRALDH1A1
SCHEMBL14907879 0.73 CYP3A4 (0.54) CA1CA2CYP3A4TSHRALDH1A1
SCHEMBL14085077 0.73 CYP3A4 (0.54) CA1CA2CYP3A4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019671-A2 BIVALENT SMAC MIMETICS AND THE USES THEREOF THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2009-02-04 EP disclosed
WO-2007130626-A2 BIVALENT SMAC MIMETICS AND THE USES THEREOF THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2007-11-15 WO disclosed