SCHEMBL4558640

SCHEMBL4558640

CCn1c(=O)n(CC(=O)O)c2c(C)ccc(C)c21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.49
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 2/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
GLA P06280 1/20 0.38
HTT P42858 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
ADORA2B P29275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30004036 0.77 APEX1 (0.52) APEX1KDM4EALDH1A1GLAADORA2B
SCHEMBL5329443 0.74 APEX1 (0.82) APEX1KDM4EALDH1A1POLBGLA
SCHEMBL3591763 0.70 KDM4E (0.42) APEX1KDM4EALDH1A1GRIN2DGRIN3B
SCHEMBL4560787 0.70 GRIN2D (0.42) APEX1KDM4EALDH1A1GRIN2DGRIN3B
SCHEMBL677187 0.70 APEX1 (0.62) APEX1KDM4EALDH1A1GLAADORA2B
SCHEMBL29251527 0.69 APEX1 (0.53) APEX1KDM4EALDH1A1GRIN2DGRIN3B
SCHEMBL12357459 0.68 APEX1 (0.41) APEX1KDM4EALDH1A1POLBMAPT
SCHEMBL12357451 0.68 APEX1 (0.44) APEX1KDM4EALDH1A1POLBMAPT
SCHEMBL3374638 0.68 APEX1 (0.65) APEX1KDM4EALDH1A1MAPTGLA
SCHEMBL24666582 0.68 KDM4E (0.44) APEX1KDM4EALDH1A1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065062-A1 NOVEL ANTIVIRAL COMPOUNDS PHARMARESOURCES(SHANGHAI)CO., LTD. (CN) 2012-05-18 WO disclosed
WO-2012065062-A1 NOVEL ANTIVIRAL COMPOUNDS PHARMARESOURCES(SHANGHAI)CO., LTD. (CN) 2012-05-18 WO disclosed