SCHEMBL4558719

SCHEMBL4558719

CSc1ccc(CSc2nc(-c3ccccc3)c(-c3ccncc3)[nH]2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.71
MAPK13 O15264 7/20 0.57
MAPK12 P53778 7/20 0.57
MAPK11 Q15759 7/20 0.57
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
PRKD3 O94806 1/20 0.50
MAP4K4 O95819 1/20 0.50
LCK P06239 1/20 0.50
RET P07949 1/20 0.50
ALOX5 P09917 1/20 0.50
PRKACA P17612 1/20 0.50
RPS6KB1 P23443 1/20 0.50
MATK P42679 1/20 0.50
FRK P42685 1/20 0.50
MAPK9 P45984 1/20 0.50
GCGR P47871 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4458847 0.89 MAPK14 (0.72) MAPK14MAPK13MAPK12MAPK11PRKD3
SCHEMBL6581827 0.89 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11PRKD3
SCHEMBL4474894 0.89 MAPK14 (0.72) MAPK14MAPK13MAPK12MAPK11PRKD3
SCHEMBL9209796 0.88 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11KDM4E
Hydrochloric Acid SCHEMBL9203423 0.86 MAPK14 (0.75) MAPK14MAPK13MAPK12MAPK11KDM4E
SCHEMBL9216064 0.85 MAPK14 (0.67) MAPK14MAPK13MAPK12MAPK11KDM4E
SCHEMBL4476561 0.83 MAPK14 (0.67) MAPK14MAPK13MAPK12MAPK11
SCHEMBL4464495 0.83 MAPK14 (0.70) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL9665340 0.82 MAPK14 (0.71) MAPK14MAPK13MAPK12MAPK11KDM4E
SCHEMBL4467677 0.81 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582660-B2 2-thio-substituted imidazole derivatives and their use in pharmaceutics C-A-I-R BIOSCIENCES GMBH (DE) 2009-09-01 US disclosed
EP-1539741-A1 2-THIO-SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR USE IN PHARMACEUTICS MERCKLE GMBH (DE) 2005-06-15 EP disclosed
WO-2004018458-A1 2-THIO-SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR USE IN PHARMACEUTICS MERCKLE-GMBH (DE) 2004-03-04 WO disclosed