SCHEMBL455875

SCHEMBL455875

NNC(=S)NC1CCc2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
MAPT P10636 1/20 0.54
ALDH1A1 P00352 3/20 0.53
PDPK1 O15530 1/20 0.53
PTPN7 P35236 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
RECQL P46063 1/20 0.48
SLC18A3 Q16572 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
TAS1R2 Q8TE23 1/20 0.46
HTT P42858 1/20 0.46
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
BCHE P06276 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
ACHE P22303 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9315471 0.81 MEN1 (0.52) MEN1KMT2AMAPTALDH1A1PDPK1
SCHEMBL11310918 0.81 PDPK1 (0.53) MEN1KMT2AALDH1A1PDPK1CA1
SCHEMBL7651926 0.80 KMT2A (0.67) MEN1KMT2AMAPTALDH1A1PDPK1
SCHEMBL3219943 0.79 ALDH1A1 (0.62) MEN1KMT2AMAPTALDH1A1PDPK1
SCHEMBL4700260 0.79 ALDH1A1 (0.62) MEN1KMT2AMAPTALDH1A1PDPK1
SCHEMBL18539280 0.77 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL1691714 0.77 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL31388654 0.77 PDPK1 (0.66) PDPK1CA1CA2SLC18A3MAOA
SCHEMBL2073072 0.77 CA1 (0.57) MEN1KMT2AMAPTALDH1A1PDPK1
SCHEMBL1441195 0.77 CA1 (0.57) MEN1KMT2AMAPTALDH1A1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101312945-A Indanyl- and tetrahydronaphtyl-amino-thiourea compounds for combating animal pests BASF SE (DE) 2008-11-26 CN claimed
WO-2012033601-A1 THIOSEMICARBAZONES WITH MDR1 - INVERSE ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2012-03-15 WO disclosed
CN-101312945-A Indanyl- and tetrahydronaphtyl-amino-thiourea compounds for combating animal pests BASF SE (DE) 2008-11-26 CN disclosed