SCHEMBL455896

SCHEMBL455896

Cc1cccc(-c2nn3ccccc3c2-c2ccc3oc(C(=O)NCCN(C)C)cc3c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.41
TGFBR1 P36897 3/20 0.40
PIK3CB P42338 1/20 0.39
HTR1A P08908 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
DRD3 P35462 1/20 0.39
MKNK1 Q9BUB5 2/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37
OPRM1 P35372 2/20 0.37
TMEM97 Q5BJF2 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
ACKR3 P25106 1/20 0.37
OPRK1 P41145 1/20 0.37
CHRM1 P11229 2/20 0.36
HPGD P15428 1/20 0.36
ALOX12 P18054 1/20 0.36
PTGER4 P35408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230400 0.87 TGFBR1 (0.36) TGFBR1PIK3CBHTR2CMKNK1ALDH1A1
SCHEMBL4868607 0.84 PIM1 (0.42) TGFBR1CHRM1TP53LMNA
SCHEMBL4868921 0.74 EGFR (0.40) CYP2D6TGFBR1ALDH1A1KDM4EHSD17B10
SCHEMBL413509 0.74 TGFBR1 (0.47) TGFBR1HPGD
SCHEMBL412319 0.74 TGFBR1 (0.61) TGFBR1PTGER4TP53
SCHEMBL412300 0.74 TGFBR1 (0.70) TGFBR1TP53
SCHEMBL4865571 0.72 BAZ2B (0.44) TGFBR1
SCHEMBL4869215 0.71 TGFBR1 (0.42) TGFBR1
SCHEMBL412491 0.70 TGFBR1 (0.57) TGFBR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL411796 0.70 TGFBR1 (0.48) TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120021519-A1 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-26 US disclosed