SCHEMBL45628

SCHEMBL45628

CC(NC1CCOCC1)c1cc(NCOCC[Si](C)(C)C)n2ncc(I)c2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 8/20 0.38
CDK9 P50750 7/20 0.38
NPY1R P25929 6/20 0.36
CDK4 P11802 3/20 0.32
CDK7 P50613 3/20 0.32
PDE4B Q07343 1/20 0.31
CCNT1 O60563 2/20 0.31
CDK1 P06493 2/20 0.31
CCNA2 P20248 2/20 0.31
CCND1 P24385 2/20 0.31
CCNE1 P24864 2/20 0.31
CCNH P51946 2/20 0.31
CCNA1 P78396 2/20 0.31
CDK3 Q00526 2/20 0.31
CDK6 Q00534 2/20 0.31
CDK5 Q00535 2/20 0.31
CDK5R1 Q15078 2/20 0.31
TTK P33981 3/20 0.31
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30638 0.83 NPY1R (0.30) NPY1R
SCHEMBL7883676 0.70 CDK2 (0.35) CDK2
SCHEMBL16104577 0.68 HSD17B10 (0.38) GSK3B
SCHEMBL588833 0.68 CCNT1 (0.39) CDK2CDK9CDK4CDK7CCNT1
SCHEMBL7874241 0.67 TTK (0.33) TTK
SCHEMBL29141 0.66 NTRK1 (0.32)
SCHEMBL45819 0.65 PDE1A (0.31) PDE1BPDE1C
SCHEMBL15026310 0.63 TTK (0.39) CDK2CDK9TTK
SCHEMBL31400 0.63 TTK (0.39) CDK2CDK9TTK
SCHEMBL7883776 0.61 NPC1 (0.36) TTKGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027234-A1 FUSED TRICYCLIC INHIBITORS OF MAMMALIAN TARGET OF RAPAMYCIN SCHERING CORPORATION (US) 2012-03-01 WO disclosed