SCHEMBL4562849

SCHEMBL4562849

O=C(c1sc2c(ccc(=O)n2-c2c(F)cccc2F)c1Br)N1CCC(O)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.34
HTR2C P28335 2/20 0.33
RAB9A P51151 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
SCN9A Q15858 2/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
SLC16A1 P53985 1/20 0.32
ADORA2A P29274 3/20 0.32
ADORA2B P29275 2/20 0.32
ADORA3 P0DMS8 1/20 0.32
PDK2 Q15119 1/20 0.32
CXCR1 P25024 1/20 0.32
CXCR2 P25025 1/20 0.32
PDE4B Q07343 1/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3118759 1.00 TYK2 (0.34) TYK2HTR2CRAB9AALOX5APFEN1
SCHEMBL3114743 1.00 TYK2 (0.34) TYK2HTR2CRAB9AALOX5APFEN1
SCHEMBL1266738 0.85 POLB (0.35) RAB9ACYP3A4SLC16A1ADORA2AADORA2B
SCHEMBL1267126 0.85 POLB (0.35) RAB9ACYP3A4SLC16A1ADORA2AADORA2B
SCHEMBL1266545 0.82 NOTUM (0.34) HTR2CRAB9ACYP3A4CYP2C9SLC16A1
SCHEMBL1266692 0.82 NOTUM (0.34) HTR2CRAB9ACYP3A4CYP2C9SLC16A1
SCHEMBL1265818 0.81 ALDH1A1 (0.36) HTR2CRAB9ACYP3A4CYP2C9SLC16A1
SCHEMBL1265514 0.81 ALDH1A1 (0.36) HTR2CRAB9ACYP3A4CYP2C9SLC16A1
SCHEMBL3113159 0.81 MAPK14 (0.33) MAPK14
SCHEMBL3113114 0.81 MAPK14 (0.33) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099805-A2 NOVEL AMINOTHIENOPYRIDINONE DERIVATIVES PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS THEREOF UCB Pharma S.A. (BE) 2009-09-16 EP claimed
WO-2008064829-A2 NOVEL AMINOTHIENOPYRIDINONE DERIVATIVES PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS THEREOF UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed