SCHEMBL4563754

SCHEMBL4563754

N#CC(F)c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
MAPT P10636 3/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 3/20 0.41
ALOX15 P16050 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 2/20 0.41
ACP3 P15309 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
S1PR2 O95136 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP3A4 P08684 2/20 0.39
CISD1 Q9NZ45 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658369 0.79 GAA (0.43) GAAMAPTALDH1A1TSHRALOX15
SCHEMBL3061003 0.78 GAA (0.42) GAAMAPTALDH1A1TSHRALOX15
SCHEMBL3556521 0.78 HDAC4 (0.42) TSHRAOC3
SCHEMBL27952753 0.77 ACP3 (0.43) GAAMAPTALDH1A1TSHRHPGD
SCHEMBL16961808 0.76 ACP3 (0.46) ALDH1A1TSHRACP3MEN1KMT2A
SCHEMBL14991566 0.76 GAA (0.41) GAAMAPTALDH1A1TSHRALOX15
SCHEMBL16321509 0.76 GAA (0.41) GAAMAPTALDH1A1TSHRALOX15
SCHEMBL5740427 0.76 OPRM1 (0.44) GAAMAPTALDH1A1TSHRALOX15
SCHEMBL6691199 0.76 TSHR (0.57) GAAMAPTALDH1A1TSHRALOX15
SCHEMBL16956469 0.76 GAA (0.41) GAAMAPTALDH1A1TSHRALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124913-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS Novartis AG (CH) 2009-12-02 EP disclosed
WO-2008077597-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS NOVARTIS AG (CH) 2008-07-03 WO disclosed
US-4369322-A WITH CYANOGEN CHLORIDE DEGUSSA AG (DE) 1983-01-18 US disclosed