SCHEMBL4563807

SCHEMBL4563807

COC(=O)c1ccc(OC(=O)c2ccc(O)cc2C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
PDK2 Q15119 1/20 0.50
PDK4 Q16654 1/20 0.50
CFTR P13569 2/20 0.43
NOTUM Q6P988 1/20 0.43
KMT2A Q03164 5/20 0.43
ESR1 P03372 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.43
NR1H4 Q96RI1 2/20 0.42
ESRRA P11474 1/20 0.42
NPC1 O15118 3/20 0.42
ESR2 Q92731 3/20 0.42
CASP3 P42574 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1940800 0.90 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL4563805 0.85 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL22979384 0.82 KDM4E (0.51) CA1CA2CFTRNOTUMESRRA
SCHEMBL34470295 0.78 EPHX2 (0.51) CA12CA1CA2CA7CA9
SCHEMBL24436898 0.77 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL3901554 0.76 CFTR (0.44) CA12CA1CA2CA7CA9
SCHEMBL696042 0.76 XDH (0.48) PDK2PDK4CFTRNOTUMMAPT
SCHEMBL28516546 0.76 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL22749359 0.75 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL12362557 0.75 CFTR (0.43) CFTRNOTUMKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118067-A1 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS Siena Biotech S.p.A. (IT) 2009-11-18 EP disclosed
WO-2008087529-A1 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS SIENA BIOTECH S.P.A. (IT) 2008-07-24 WO disclosed