SCHEMBL4565058

SCHEMBL4565058

C=Cc1cc2c(OC3C[C@@H](C(=O)O)N(C(C)=O)C3)nccc2cc1OC

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.38
ANPEP P15144 1/20 0.38
STING1 Q86WV6 1/20 0.37
CYP3A4 P08684 1/20 0.36
PIK3CD O00329 2/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 2/20 0.35
IRAK4 Q9NWZ3 12/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4297033 0.94 STING1 (0.38) STING1CYP3A4IRAK4
SCHEMBL1074488 0.89 CYP3A4 (0.40) STING1CYP3A4PIK3CDPIK3CAPIK3CB
SCHEMBL1074490 0.89 CYP3A4 (0.40) STING1CYP3A4PIK3CDPIK3CAPIK3CB
Hydrochloric Acid SCHEMBL1071141 0.86 IRAK4 (0.39) STING1IRAK4
SCHEMBL16318483 0.82 CYP3A4 (0.41) MMP2ANPEPCYP3A4PIK3CDPIK3CA
SCHEMBL16318484 0.82 CYP3A4 (0.41) MMP2ANPEPCYP3A4PIK3CDPIK3CA
SCHEMBL4301154 0.80 APAF1 (0.39) CYP3A4IRAK4
SCHEMBL4298045 0.79 CYP3A4 (0.38) CYP3A4IRAK4
SCHEMBL12934494 0.78 CYP3A4 (0.38) CYP3A4PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16318497 0.78 CYP3A4 (0.55) CYP3A4IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079479-A2 HCV NS3 PROTEASE INHIBITORS Merck & Co., Inc. (US) 2009-07-22 EP disclosed
WO-2008051475-A2 HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2008-05-02 WO disclosed