SCHEMBL4565285

SCHEMBL4565285

Cc1cc(C(=O)O)cc2nc(C3CCCO3)[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FASN P49327 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.36
HNF4A P41235 1/20 0.35
PTGES O14684 2/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
PTGER4 P35408 1/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 1/20 0.34
TYK2 P29597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565286 0.83 FASN (0.37) FASNPTGESKDM4EALDH1A1HSD17B10
SCHEMBL13907875 0.82 ALDH1A1 (0.39) FASNTSHRHTTKDM4EALDH1A1
SCHEMBL13906625 0.81 NPC1 (0.37) L3MBTL1ALDH1A1
SCHEMBL15554717 0.75 FASN (0.54) FASNL3MBTL1HNF4ATSHRHTT
SCHEMBL13907803 0.72 TDP1 (0.53) TSHRKDM4EALDH1A1HSD17B10HPGD
SCHEMBL13907999 0.70 KMT2A (0.39) FASNALDH1A1HSD17B10
SCHEMBL15554667 0.69 FASN (0.47) FASNPTGES
SCHEMBL13906484 0.68 NPY5R (0.43) L3MBTL1TSHRHTTKDM4EALDH1A1
SCHEMBL8847760 0.67 ADORA1 (0.46) TSHRHTTKDM4EALDH1A1HPGD
SCHEMBL31401543 0.67 TSHR (0.52) HNF4ATSHRHTTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed