SCHEMBL4565318

SCHEMBL4565318

CCn1c(=O)c(-c2cncnc2)cc2c(C)nc(NS(=O)(=O)CC)nc21

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
HSD17B10 Q99714 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
PIK3CA P42336 15/20 0.41
PIK3CD O00329 1/20 0.40
PIK3CB P42338 1/20 0.40
MTOR P42345 1/20 0.40
PIK3CG P48736 1/20 0.40
PDE4B Q07343 1/20 0.35
PDE7A Q13946 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL189119 0.86 ALDH1A1 (0.64) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL1901551 0.80 PIK3CA (0.60) PIK3CAPIK3CDPIK3CBMTORPIK3CG
SCHEMBL189326 0.71 ALDH1A1 (0.65) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL15146960 0.70 PIK3CA (0.54) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL189165 0.70 FGFR1 (0.51) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL4231600 0.70 ADORA1 (0.46) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL188797 0.70 ALDH1A1 (0.63) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL15109485 0.70 PIK3CA (0.51) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL188738 0.70 HSD17B10 (0.63) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL189369 0.70 ALDH1A1 (0.63) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065019-A2 PYRIDOPYRIMIDINONE INHIBITORS OF P13K ALPHA EXELIXIS, INC. (US) 2012-05-18 WO disclosed