SCHEMBL4565597

SCHEMBL4565597

Cc1cnc(CN(Cc2ncccc2C(C)C)C2CCCCN2C(=O)Nc2cccnn2)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 3/20 0.35
PRMT5 O14744 2/20 0.33
WDR77 Q9BQA1 2/20 0.33
TRPV1 Q8NER1 1/20 0.32
MAPT P10636 1/20 0.32
FAAH O00519 5/20 0.31
BTK Q06187 3/20 0.31
SMO Q99835 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2085997 0.85 GSK3B (0.36) CXCR4TRPV1FAAH
SCHEMBL2084436 0.78 FAAH (0.38) CXCR4TRPV1FAAH
SCHEMBL2082165 0.75 GSK3B (0.35) CXCR4TRPV1
SCHEMBL12935463 0.75 TRPV1 (0.34) CXCR4TRPV1
SCHEMBL2084022 0.74 CXCR4 (0.38) CXCR4TRPV1MAPTSMO
SCHEMBL23428604 0.74 CXCR4 (0.46) CXCR4MAPTBTK
SCHEMBL2083283 0.74 CXCR4 (0.39) CXCR4TRPV1MAPTSMO
SCHEMBL5058354 0.73 CXCR4 (0.39) CXCR4MAPT
SCHEMBL2083906 0.73 CXCR4 (0.36) CXCR4TRPV1MAPTSMO
SCHEMBL2083541 0.72 CXCR4 (0.40) CXCR4TRPV1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed