SCHEMBL4566137

SCHEMBL4566137

O=C(OCc1ccc(-c2cc3cc(Cc4ccccc4)ccc3o2)cc1)C1CCNCC1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 10/20 0.58
S1PR3 Q99500 3/20 0.50
FFAR1 O14842 2/20 0.46
KCNH2 Q12809 1/20 0.46
TSHR P16473 1/20 0.42
MAOB P27338 2/20 0.40
MAP2K1 Q02750 1/20 0.39
HRH1 P35367 1/20 0.39
KDM5A P29375 1/20 0.39
F10 P00742 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5063301 0.83 S1PR1 (0.58) S1PR1S1PR3FFAR1MAOB
SCHEMBL606466 0.78 TSHR (0.55) TSHR
Hydrochloric Acid SCHEMBL3494457 0.77 TSHR (0.57) TSHR
SCHEMBL1602267 0.74 S1PR1 (0.81) S1PR1S1PR3FFAR1KCNH2MAOB
SCHEMBL1603237 0.73 S1PR1 (1.00) S1PR1S1PR3KCNH2
Alcohol SCHEMBL27541427 0.73 TSHR (0.53) TSHRF10
SCHEMBL28687641 0.73 TSHR (0.53) TSHRF10
SCHEMBL1601401 0.73 S1PR1 (0.52) S1PR1S1PR3FFAR1KCNH2MAOB
SCHEMBL1602885 0.71 S1PR1 (0.58) S1PR1S1PR3FFAR1KCNH2MAOB
SCHEMBL3699394 0.71 MAOB (0.63) S1PR1S1PR3FFAR1KCNH2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1965807-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF Epix Delaware, Inc. (US) 2008-09-10 EP claimed
WO-2007061458-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-05-31 WO claimed
EP-2364976-B1 S1P receptor modulating compounds and use thereof EPIX PHARM INC (US) 2014-10-08 EP disclosed
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP disclosed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed