SCHEMBL5063301

SCHEMBL5063301

CCCCc1ccc2oc(-c3ccc(COC(=O)C4CCNCC4)cc3)cc2c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.58
ACHE P22303 3/20 0.45
FFAR1 O14842 2/20 0.43
MAOB P27338 3/20 0.41
S1PR3 Q99500 2/20 0.41
CYP2C8 P10632 1/20 0.41
ALOX5 P09917 2/20 0.38
PTGES O14684 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4566137 0.83 S1PR1 (0.58) S1PR1FFAR1MAOBS1PR3
SCHEMBL1601906 0.74 S1PR1 (0.82) S1PR1FFAR1S1PR3
SCHEMBL1600903 0.73 S1PR1 (1.00) S1PR1S1PR3
SCHEMBL1602093 0.71 S1PR1 (0.57) S1PR1ACHEFFAR1MAOBCYP2C8
SCHEMBL3812511 0.69 S1PR1 (0.69) S1PR1ACHEFFAR1S1PR3CYP2C8
Alcohol SCHEMBL27541427 0.68 TSHR (0.53)
SCHEMBL12706849 0.68 S1PR1 (0.69) S1PR1ACHEMAOBS1PR3CYP2C8
SCHEMBL28202643 0.68 FABP7 (0.50)
SCHEMBL606466 0.67 TSHR (0.55)
SCHEMBL7601727 0.66 RARB (0.61) S1PR1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1965807-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF Epix Delaware, Inc. (US) 2008-09-10 EP claimed
WO-2007061458-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-05-31 WO claimed
EP-1965807-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF Epix Delaware, Inc. (US) 2008-09-10 EP disclosed
WO-2007061458-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-05-31 WO disclosed