SCHEMBL4566146

SCHEMBL4566146

COc1ccc(C(C)CC(N)=O)nc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.41
TNF P01375 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
PARP10 Q53GL7 2/20 0.39
PARP1 P09874 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
PARP4 Q9UKK3 1/20 0.39
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
HPGDS O60760 4/20 0.38
ACACB O00763 1/20 0.37
VNN1 O95497 1/20 0.36
APLNR P35414 2/20 0.36
DCAF1 Q9Y4B6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1871235 0.82 CACNA1I (0.53) CACNA1IL3MBTL1
SCHEMBL19738832 0.80 CACNA1I (0.46) CACNA1ICA1CA2PARP10PARP1
SCHEMBL29376832 0.80 CACNA1I (0.46) CACNA1ICA1CA2PARP10PARP1
SCHEMBL3728573 0.78 APLNR (0.50) APLNR
SCHEMBL19716796 0.78 CACNA1I (0.44) CACNA1ICA1CA2PARP10PARP1
SCHEMBL19464658 0.77 CACNA1I (0.43) CACNA1ICA1CA2GAAAPLNR
SCHEMBL27692987 0.76 CACNA1I (0.48) CACNA1ICA1CA2HTTHPGDS
SCHEMBL12883281 0.76 TNF (0.54) L3MBTL1TNFCA1CA2PARP10
SCHEMBL1063334 0.73 CACNA1I (0.42) CACNA1ICA1CA2
SCHEMBL14864691 0.73 CACNA1I (0.48) CACNA1ICA1CA2ACACBAPLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010493-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120729-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-10-25 WO disclosed