SCHEMBL4566147

SCHEMBL4566147

COc1ccc(C(C)NC(C)=O)nc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 2/20 0.60
ACACB O00763 10/20 0.51
PPARD Q03181 1/20 0.45
PPARA Q07869 1/20 0.45
ACACA Q13085 1/20 0.44
CACNA1G O43497 1/20 0.44
CACNA1H O95180 1/20 0.44
CNR2 P34972 1/20 0.44
KCNH2 Q12809 1/20 0.44
MTNR1A P48039 3/20 0.43
MTNR1B P49286 3/20 0.43
CNR1 P21554 1/20 0.43
HPGDS O60760 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21920417 0.82 CACNA1I (0.65) CACNA1IACACBACACACACNA1GCACNA1H
Hydrochloric Acid SCHEMBL29791928 0.79 CACNA1I (0.67) CACNA1IACACBACACACACNA1GCACNA1H
SCHEMBL15022712 0.79 ESR1 (0.46) CACNA1IACACBPPARDPPARAACACA
SCHEMBL15022711 0.79 ESR1 (0.46) CACNA1IACACBPPARDPPARAACACA
SCHEMBL2134729 0.78 CACNA1I (0.73) CACNA1ICNR1HPGDS
SCHEMBL2134726 0.78 CACNA1I (0.73) CACNA1ICNR1HPGDS
SCHEMBL588472 0.78 APLNR (0.48) CACNA1IACACBACACACACNA1GCACNA1H
SCHEMBL588802 0.78 B3GNT2 (0.47) CACNA1IACACB
SCHEMBL12069877 0.78 APLNR (0.48) CACNA1IACACBACACACACNA1GCACNA1H
SCHEMBL588473 0.78 APLNR (0.48) CACNA1IACACBACACACACNA1GCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010493-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120729-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-10-25 WO disclosed