SCHEMBL4570634

SCHEMBL4570634

Cc1cccc(C(=O)c2c[nH]c3ncc(Br)cc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.47
BRD4 O60885 2/20 0.46
BRAF P15056 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CDK2 P24941 2/20 0.44
PLK4 O00444 1/20 0.44
AURKA O14965 1/20 0.44
JAK2 O60674 1/20 0.44
ROCK2 O75116 1/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
PRKCG P05129 1/20 0.44
INSR P06213 1/20 0.44
CDK1 P06493 1/20 0.44
FES P07332 1/20 0.44
IGF1R P08069 1/20 0.44
ROS1 P08922 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL856914 0.86 BRAF (0.46) AAK1BRD4BRAFCDK2PLK4
SCHEMBL1363568 0.86 AAK1 (0.58) AAK1BRD4BRAFHTTCDK2
SCHEMBL4570635 0.85 AAK1 (0.47) AAK1BRD4BRAFALDH1A1HPGD
SCHEMBL858197 0.85 BRAF (0.53) AAK1BRD4BRAFCDK2PLK4
SCHEMBL4570622 0.85 BRAF (0.49) AAK1BRD4BRAFALDH1A1HPGD
SCHEMBL3506984 0.85 AXL (0.50) AAK1BRD4BRAFCDK2PLK4
SCHEMBL297306 0.85 BRAF (0.45) AAK1BRD4BRAFCDK2PLK4
SCHEMBL857107 0.85 AAK1 (0.53) AAK1BRAFROCK2PRKD3MAP4K4
SCHEMBL411351 0.82 BRD4 (0.48) AAK1BRD4BRAFNPSR1CDK2
SCHEMBL21624518 0.81 KMT2A (0.49) AAK1BRAFALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120122860-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122860-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS BRAF, RAF1, ARAF AAK1 247/4885BRD4 2367/4885BRAF 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.