SCHEMBL4570635

SCHEMBL4570635

Cc1cccc(C(=O)c2c[nH]c3ncc(F)cc23)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.47
CYP3A4 P08684 1/20 0.46
BRD4 O60885 2/20 0.46
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
POLB P06746 1/20 0.44
PAK1 Q13153 2/20 0.43
CCNE2 O96020 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 2/20 0.42
BRAF P15056 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
AXL P30530 2/20 0.42
VNN1 O95497 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3705389 0.85 NEK2 (0.50) AAK1CYP3A4BRD4PAK1CDK2
SCHEMBL4570634 0.85 AAK1 (0.47) AAK1BRD4ALDH1A1HPGDHTT
SCHEMBL297839 0.85 AAK1 (0.45) AAK1CYP3A4BRD4POLBPAK1
SCHEMBL4570622 0.85 BRAF (0.49) AAK1CYP3A4BRD4ALDH1A1HPGD
SCHEMBL415959 0.79 RIPK1 (0.60) AAK1AXL
SCHEMBL4570621 0.78 PAK1 (0.57) AAK1BRD4PAK1
SCHEMBL3710853 0.78 NEK2 (0.50) AAK1CYP3A4BRD4PAK1CDK2
SCHEMBL3705033 0.78 AAK1 (0.47) AAK1CYP3A4BRD4POLBPAK1
SCHEMBL858197 0.78 BRAF (0.53) AAK1CYP3A4BRD4PAK1CDK2
SCHEMBL4570626 0.77 CAMKK2 (0.61) AAK1CYP3A4BRD4PAK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120122860-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122860-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS BRAF, RAF1, ARAF AAK1 247/4885CYP3A4 3611/4885BRD4 2367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.