SCHEMBL4573292

SCHEMBL4573292

CC(C)(C(N)=O)c1ccc(N2CCNCC2)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 6/20 0.54
PIM1 P11309 3/20 0.46
PIM3 Q86V86 2/20 0.46
HTR3E A5X5Y0 2/20 0.46
HTR3B O95264 2/20 0.46
HTR3A P46098 2/20 0.46
HTR3D Q70Z44 2/20 0.46
HTR3C Q8WXA8 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
HTR1A P08908 1/20 0.46
CYP2D6 P10635 1/20 0.46
THRB P10828 1/20 0.46
CYP2C9 P11712 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
SLC6A4 P31645 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573342 0.85 ADRB1 (0.55) ADRB1PIM1PIM3HTR3EHTR3B
SCHEMBL4573825 0.82 ACVR1 (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL26074538 0.82 ADRB1 (0.65) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4541552 0.77 ADRB1 (0.50) ADRB1PIM1PIM3HTR3EHTR3B
SCHEMBL1471288 0.76 ADRB1 (0.65) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4573471 0.76 ADRB1 (0.56) ADRB1PIM1HTR3EHTR3BHTR3A
SCHEMBL4939443 0.73 ADRB1 (0.61) ADRB1HTR3EHTR3BHTR3AHTR3D
Tert-Butyl Formate SCHEMBL27925832 0.72 ADRB1 (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2984679 0.72 ADRB1 (0.73) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL14080465 0.72 ADRB1 (0.63) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed