SCHEMBL4573323

SCHEMBL4573323

O=S(=O)(Nc1[c]cccc1F)C1CC1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
HDAC4 P56524 1/20 0.35
SCN9A Q15858 1/20 0.35
MAP2K4 P45985 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
MAP2K7 O14733 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KIT P10721 2/20 0.33
MRGPRX1 Q96LB2 3/20 0.32
CKS1B P61024 2/20 0.32
SKP2 Q13309 2/20 0.32
HSD17B1 P14061 2/20 0.31
HSD17B2 P37059 2/20 0.31
BRPF1 P55201 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14831080 0.75 SCN9A (0.43) PTGS1PTGS2HDAC4SCN9AMAP2K4
SCHEMBL14830870 0.73 PSIP1 (0.53) PTGS1PTGS2ALOX5APFEN1MRGPRX1
SCHEMBL3648948 0.71 HDAC4 (0.40) PTGS1PTGS2HDAC4MAP2K4ALOX5AP
SCHEMBL22608 0.68
SCHEMBL4573131 0.68 PTGS1 (0.37) PTGS1PTGS2HDAC4SCN9AMAP2K4
SCHEMBL19991847 0.67 SGK1 (0.34) MAP2K4MAP2K7TDP1MRGPRX1
SCHEMBL4573296 0.67 HDAC4 (0.43) PTGS1PTGS2HDAC4MAP2K4MAP2K7
SCHEMBL1267271 0.66 BRD4 (0.40) PTGS1PTGS2HDAC4MAP2K4ALOX5AP
SCHEMBL4600157 0.65
SCHEMBL1099375 0.65 HDAC4 (0.47) PTGS1PTGS2HDAC4MAP2K4MAP2K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008077651-A1 PYRIDO(3,2-D)PYRIMIDINES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-07-03 WO claimed
WO-2008077651-A1 PYRIDO(3,2-D)PYRIMIDINES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-07-03 WO disclosed