SCHEMBL4573366

SCHEMBL4573366

COc1cccc(N2CCN(C(=O)OC(C)(C)C)C(C)C2)n1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.60
CHRM4 P08173 1/20 0.54
HDAC1 Q13547 1/20 0.50
SUV39H2 Q9H5I1 2/20 0.46
GPR119 Q8TDV5 2/20 0.46
GRM1 Q13255 5/20 0.45
HRH3 Q9Y5N1 1/20 0.44
ACACB O00763 1/20 0.42
NR1H2 P55055 3/20 0.42
NR1H3 Q13133 2/20 0.42
ALOX5 P09917 1/20 0.41
FAAH O00519 1/20 0.40
HTR1A P08908 1/20 0.40
HTR2A P28223 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116230 1.00 MAP4K4 (0.60) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL31383652 0.88 MAP4K4 (0.58) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL31383595 0.88 MAP4K4 (0.58) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL29053096 0.86 MAP4K4 (0.59) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL29053095 0.86 MAP4K4 (0.59) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL4573088 0.85 CHRM4 (0.58) MAP4K4CHRM4GRM1HRH3ACACB
SCHEMBL4584408 0.84 MAP4K4 (0.52) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL8113244 0.84 MAP4K4 (0.52) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL31383697 0.83 MAP4K4 (0.56) MAP4K4CHRM4HDAC1SUV39H2GPR119
SCHEMBL31383568 0.83 MAP4K4 (0.56) MAP4K4CHRM4HDAC1SUV39H2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed