SCHEMBL457397

SCHEMBL457397

COCCn1c(-c2ccccc2)ncc(C(=O)C2=C(O)C3CCC(C3)C2=O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.39
CYP1A2 P05177 9/20 0.39
HSD17B10 Q99714 7/20 0.39
HPGD P15428 4/20 0.38
RXFP1 Q9HBX9 1/20 0.38
BRD4 O60885 1/20 0.37
HSP90AA1 P07900 1/20 0.36
RAB9A P51151 1/20 0.36
CYP3A4 P08684 6/20 0.36
CYP2C9 P11712 6/20 0.36
LMNA P02545 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
TSHR P16473 5/20 0.35
CASP1 P29466 5/20 0.35
CASP7 P55210 5/20 0.35
CYP2C19 P33261 3/20 0.35
HIF1A Q16665 3/20 0.35
GLA P06280 2/20 0.35
CYP2D6 P10635 2/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL454637 0.87 CYP1A2 (0.40) ALDH1A1CYP1A2HSD17B10HPGDBRD4
SCHEMBL457304 0.74 TDP1 (0.39) ALDH1A1CYP1A2HSD17B10HPGDRXFP1
SCHEMBL9903971 0.69 CYP1A2 (0.40) ALDH1A1CYP1A2HSD17B10HPGDBRD4
SCHEMBL454628 0.67 SMN1; SMN2 (0.36) ALDH1A1CYP1A2HSD17B10HPGDRAB9A
SCHEMBL16435041 0.67 KMT2A (0.36) ALDH1A1RXFP1TDP1MEN1KMT2A
SCHEMBL455164 0.67 SMN1; SMN2 (0.36) ALDH1A1HSD17B10HPGDRAB9AMAPT
SCHEMBL9895278 0.66 ALDH1A1 (0.46) ALDH1A1CYP1A2HSD17B10HPGDRXFP1
SCHEMBL12487741 0.66 SMN1; SMN2 (0.35) ALDH1A1CYP1A2HSD17B10HPGDRAB9A
SCHEMBL454865 0.65 BUB1 (0.38) ALDH1A1HSD17B10HPGDBRD4RAB9A
SCHEMBL9895127 0.65 CYP1A2 (0.47) ALDH1A1CYP1A2HSD17B10HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033548-A2 HERBICIDAL BIS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-15 WO claimed
WO-2012033548-A2 HERBICIDAL BIS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-15 WO disclosed