SCHEMBL4580382

SCHEMBL4580382

COc1ccc(CNc2nccc(N3CCNC(=O)C3c3ccccc3)n2)c(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.45
TSHR P16473 8/20 0.45
CYP1A2 P05177 7/20 0.43
CYP3A4 P08684 7/20 0.43
CYP2D6 P10635 6/20 0.43
CYP2C19 P33261 6/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
USP2 O75604 3/20 0.43
KDM4E B2RXH2 4/20 0.42
LMNA P02545 4/20 0.41
CLK4 Q9HAZ1 4/20 0.41
GLA P06280 2/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
ALOX15 P16050 2/20 0.40
RECQL P46063 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4580579 0.87 ACHE (0.47) CLK4
SCHEMBL4581286 0.87 IDH1 (0.41) ALDH1A1KDM4EGAA
SCHEMBL4580743 0.81 KDR (0.50) ALDH1A1MEN1KMT2AUSP2KDM4E
SCHEMBL4581206 0.81 CYP1A2 (0.48) ALDH1A1TSHRCYP1A2CYP3A4CYP2D6
SCHEMBL4579436 0.81 FLT1 (0.52) ALDH1A1TSHRCYP1A2CYP3A4CYP2C19
SCHEMBL4581890 0.81 IDH1 (0.54)
SCHEMBL4581947 0.81 OGA (0.43) KDM4E
SCHEMBL4581037 0.80 MKNK1 (0.48)
SCHEMBL4579971 0.80 KDM4E (0.42) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4581479 0.80 IDH1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US claimed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US claimed
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US disclosed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080258-A1 Pyridine and pyrimidine derivatives ROR1, MAPK1, IRAK1 ALDH1A1 682/4885TSHR 790/4885CYP1A2 1524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.