SCHEMBL4581429

SCHEMBL4581429

O=C(O)C(=O)C(C(=O)c1cccs1)C(=O)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
DAO P14920 1/20 0.44
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
KEAP1 Q14145 1/20 0.44
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
HPGDS O60760 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
RAB9A P51151 5/20 0.39
NPC1 O15118 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
POLB P06746 2/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2802204 0.83 TSHR (0.50) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL1681118 0.79 TSHR (0.51) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL28376224 0.78 TSHR (0.50) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL5873224 0.76 TSHR (0.49) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL3249145 0.76 CYP2C9 (0.52) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL10628291 0.75 TSHR (0.48) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL5873170 0.74 CYP2C19 (0.47) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL27427456 0.73 CYP2C9 (0.49) CYP2C9CYP2C19CYP2D6TSHRDAO
SCHEMBL6135938 0.70 CYP2C19 (0.46) CYP2C9CYP2C19CYP2D6TSHRDAO
Thiophene Carboxylic Acid SCHEMBL4617799 0.70 DAO (0.76) CYP2C9CYP2C19CYP2D6TSHRDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817281-B1 Organic electroluminescent device with an inorganic electron-conducting layer PHILIPS INTELLECTUAL PROPERTY (DE) 2008-10-15 EP disclosed
EP-0697744-B1 Organic electroluminescent device PHILIPS PATENTVERWALTUNG (DE) 2000-01-05 EP disclosed
EP-0817281-A2 Organic electroluminescent device with an inorganic electron-conducting layer Philips Patentverwaltung GmbH (DE) 1998-01-07 EP disclosed
EP-0697744-A1 Organic electroluminescent device Philips Patentverwaltung GmbH (DE) 1996-02-21 EP disclosed