SCHEMBL458181

SCHEMBL458181

CC(C)(C)OC(=O)N[C@H]1CN(c2ncc(OCCC3CCN(C(=O)OCc4ccccc4)CC3)cn2)C[C@@H]1c1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.43
GRIN2B Q13224 8/20 0.40
CYP2D6 P10635 4/20 0.39
CYP2C9 P11712 4/20 0.39
CYP3A4 P08684 3/20 0.39
GPR119 Q8TDV5 5/20 0.39
FAAH O00519 1/20 0.38
YAP1 P46937 1/20 0.38
RORC P51449 2/20 0.37
CHRM4 P08173 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459391 0.93 PDE4B (0.42) PDE4BGRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL457195 0.91 PDE4B (0.42) PDE4BGRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL458155 0.87 PDE4B (0.43) PDE4BGRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL12064782 0.82 PDE4B (0.42) PDE4BGPR119YAP1RORC
SCHEMBL12064593 0.81 PDE4B (0.42) PDE4BGRIN2BGPR119YAP1RORC
SCHEMBL14730220 0.81 TP53 (0.45) PDE4BRORCCHRM4
SCHEMBL470782 0.80 PDE4B (0.42) PDE4BGRIN2BRORC
SCHEMBL150998 0.78 GPR119 (0.48) GPR119CHRM4
SCHEMBL1720991 0.78 GPR119 (0.48) GPR119CHRM4
SCHEMBL14722527 0.78 PDE4B (0.41) PDE4BGPR119RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147951-A1 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS PROSIDION LIMITED (GB) 2011-12-01 WO disclosed